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Bioorganic Chemistry|April 26, 2020
Privileged scaffold inspired design of novel oxime-biphenyl-DAPYs in treatment of HIV-1Yang Yang, Christophe Pannecouque, Erik De Clercq, et al.Bioorganic Chemistry|April 26, 2020
Fluorinated CRA13 analogues: Synthesis, in vitro evaluation, radiosynthesis, in silico and in vivo PET studyAhmed H E Hassan, Kyung Tae Park, Hye Jin Kim, et al.Bioorganic Chemistry|April 26, 2020
Identification of rapid access to polycyclic systems via a base-catalyzed cascade cyclization reaction and their biological evaluationTaotao Ling, Victor Hadi, John Bollinger, et al.Bioorganic Chemistry|April 26, 2020
Discovery of diaminopyrimidine-carboxamide derivatives as JAK3 inhibitorsRajesh Bahekar, Nandini Panchal, Shubhangi Soman, et al.Bioorganic Chemistry|April 29, 2020
Synthesis and anticancer evaluation of novel 1H-benzo[d]imidazole derivatives of dehydroabietic acid as PI3Kα inhibitorsYa-Qun Yang, Hao Chen, Qing-Song Liu, et al.Bioorganic Chemistry|May 4, 2020
Design, synthesis, and pharmacological evaluation of novel and selective COX-2 inhibitors based on bumetanide scaffoldTarek S Ibrahim, Ibrahim M Salem, Samia M Mostafa, et al.Bioorganic Chemistry|April 13, 2020
In vivo efficacy studies of novel quinazoline derivatives as irreversible dual EGFR/HER2 inhibitors, in lung cancer xenografts (NCI-H1975) mice modelsDebasis Das, Lingzhi Xie, Jingbing Wang, et al.Bioorganic Chemistry|May 1, 2020
Synthesis and evaluation of new 1,2,4-oxadiazole based trans- acrylic acid derivatives as potential PPAR-alpha/gamma dual agonistParanjeet Kaur, Zahid Rafiq Bhat, Sana Bhat, et al.Bioorganic Chemistry|May 4, 2020
An okadaic acid fragment analogue prevents nicotine-induced resistance to cisplatin by recovering PP2A activity in non-small cell lung cancer cellsRaquel L Arribas, Anna Bordas, Judit Domènech Omella, et al.Bioorganic Chemistry|May 4, 2020
Design, synthesis, in vitro and in silico studies of 2, 3-diaryl benzofuran derivatives as antitubercular agentsBalakishan Bhukya, Aparna Shukla, Vinita Chaturvedi, et al.Pageof 868