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Bioorganic Chemistry|November 25, 2020
In silico designing, in vitro and in vivo evaluation of potential PPAR-γ agonists derived from aryl propionic acid scaffoldChetna Kharbanda, Mohammad Sarwar Alam, Hinna Hamid, et al.Bioorganic Chemistry|November 28, 2020
Targeting and imaging of HER2 overexpression tumor with a new peptide-based 68Ga-PET radiotracerJavad Biabani Ardakani, Mehdi Akhlaghi, Babak Nikkholgh, et al.Bioorganic Chemistry|November 28, 2020
The relationship between stereochemical and both, pharmacological and ADME-Tox, properties of the potent hydantoin 5-HT7R antagonist MF-8Katarzyna Kucwaj-Brysz, Gniewomir Latacz, Sabina Podlewska, et al.Bioorganic Chemistry|September 5, 2020
Capsaicin: A "hot" KDM1A/LSD1 inhibitor from peppersGang Jia, Shundong Cang, Peizhi Ma, et al.Bioorganic Chemistry|September 5, 2020
Design, synthesis, biological evaluation, and docking study of novel dual-acting thiazole-pyridiniums inhibiting acetylcholinesterase and β-amyloid aggregation for Alzheimer's diseaseGolaleh Ghotbi, Mohammad Mahdavi, Zahra Najafi, et al.Bioorganic Chemistry|September 5, 2020
Novel CoFe2O4@ZnO-CeO2 ternary nanocomposite: Sonochemical green synthesis using Crataegus microphylla extract, characterization and their application in catalytic and antibacterial activitiesAli Naghizadeh, Sarvin Mohammadi-Aghdam, Sobhan Mortazavi-DerazkolaBioorganic Chemistry|September 5, 2020
NQO1-selective activated prodrugs of combretastatin A-4: Synthesis and biological evaluationChong Zhang, Yan Qu, Xin Ma, et al.Bioorganic Chemistry|September 5, 2020
Structurally diverse sesquiterpenoids from the aerial parts of Artemisia annua (Qinghao) and their striking systemically anti-inflammatory activitiesDa-Peng Qin, Hai-Bo Li, Qian-Qian Pang, et al.Bioorganic Chemistry|September 5, 2020
Evaluation of anti rheumatic activity of Piper betle L. (Betelvine) extract using in silico, in vitro and in vivo approachesSelvakumar Murugesan, Devibala Ravichandran, Dinesh Kumar Lakshmanan, et al.Bioorganic Chemistry|September 6, 2020
Synthesis of nitrogen, phosphorus, selenium and sulfur-containing heterocyclic compounds - Determination of their carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase and α-glycosidase inhibition propertiesİlhami Gülçin, Boris Trofimov, Ruya Kaya, et al.Pageof 868