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Bioorganic Chemistry|April 23, 2024
Synthesis and biological evaluation of Halogen-Substituted novel α-Ketoamides as potential protein aggregation modulators in Alzheimer's diseaseBhanuranjan Das, Anurag Tk Baidya, Sourabh Chakrabarti, et al.Bioorganic Chemistry|April 23, 2024
Lathyrane and premyrsinane Euphorbia diterpenes against Alzheimer's disease: Bioinspired synthesis, anti-cholinesterase and neuroprotection bioactivityLian Sun, Xin-Ming Wang, Qianhui Tang, et al.Bioorganic Chemistry|April 25, 2024
Synthesis and evaluation of pentacyclic triterpenoids conjugates as novel HBV entry inhibitors targeting NTCP receptorYixin Chen, Meitao Duan, Xiangwan Wang, et al.Bioorganic Chemistry|April 11, 2024
Development of D-π-A organic dyes for discriminating HSA from BSA and study on dye-HSA interactionHao-Wen Cao, Yan-Song Chen, Jing-Zhi Li, et al.Bioorganic Chemistry|April 10, 2024
Discovery of PXR agonists from Hypericum japonicum: A class of novel nonaromatic acylphloroglucinol-terpenoid adductsHaiguo Su, Hangfei Liang, Jianing Tian, et al.Bioorganic Chemistry|April 11, 2024
d-type peptides based fluorescent probes for "turn on" sensing of heparinHuan Xu, Xing-Yan Fu, Yong-Xin Bao, et al.Bioorganic Chemistry|April 11, 2024
Rapid identifying of COX-2 inhibitors from turmeric (Curcuma longa) by bioaffinity ultrafiltration coupled with UPLC-Q Exactive-Orbitrap-MS and zebrafish-based in vivo validationZhenwei Lan, Rui Yang, Hu Wang, et al.Bioorganic Chemistry|April 13, 2024
Discovery of a new class of potent pyrrolo[3,4-c]quinoline-1,3-diones based inhibitors of human dihydroorotate dehydrogenase: Synthesis, pharmacological and toxicological evaluationMarina G Dimitrijević, Cornelia Roschger, Kevin Lang, et al.Bioorganic Chemistry|January 23, 2026
Toward multi-target therapy: Design, synthesis and mechanistic profiling of some novel acyl-thiosemicarbazides, as MAO and aromatase inhibitorsAhmet Avci, Hayrünnisa Taşci, Begüm Nurpelin Sağlık Özkan, et al.Bioorganic Chemistry|January 27, 2026
Triazinyl-benzenesulfonamide derivatives as hCA IX inhibitors: Design, synthesis, and activity determination using an optimized stop-flow methodologyVojtech Varecka, Karolina Seligova, Alena Hofrova, et al.Pageof 868