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Bioorganic Chemistry|April 6, 2024
Bioisosteric replacement strategy leads to novel DNA gyrase B inhibitors with improved potencies and propertiesWenjie Xue, Xueping Zuo, Xueqi Zhao, et al.Bioorganic Chemistry|April 7, 2024
Novel partially reversible NDM-1 inhibitors based on the naturally occurring houttuyninLifang Wang, Yaowen Liang, Pan Luo, et al.Bioorganic Chemistry|April 5, 2024
Discovery of a novel small-molecule activator of SIRT3 that inhibits cell proliferation and migration by apoptosis and autophagy-dependent cell death pathways in colorectal cancerYi Mou, Yanmei Chen, Zhichao Fan, et al.Bioorganic Chemistry|April 3, 2024
A novel natural Syk inhibitor suppresses IgE-mediated mast cell activation and passive cutaneous anaphylaxisLele Wang, Yuzhen Fang, Yuqing Ma, et al.Bioorganic Chemistry|March 26, 2024
Discovery of cinnamylaldehyde-derived mono-carbonyl curcumin analogs as anti-gastric cancer agents via suppression of STAT3 and AKT pathwayXi Chen, Peiqin Zhang, Huating Zhang, et al.Bioorganic Chemistry|March 24, 2024
2,3-Dichloronaphthoquinone derivatives: Synthesis, antimicrobial activity, molecular modelling and ADMET studiesHakan Kolancılar, Hafize Özcan, Ayşen Şuekinci Yılmaz, et al.Bioorganic Chemistry|March 26, 2024
Discovery of sesquiterpenoids from an actinomycete Crossiella cryophila through genome mining and heterologous expressionQian Yang, Jupeng Tian, Shungen Chen, et al.Bioorganic Chemistry|March 25, 2024
Accurate detection depression cell model with a dual-locked fluorescence probe in response to noradrenaline and HClOXinyi Xiong, Jianwen Qiu, Shaofei Fu, et al.Bioorganic Chemistry|March 17, 2024
Four component Ugi reaction based small-molecule probes for integrated phenotypic screeningManikandan Thangaraj, Ksenia Lialin, Rambabu Dandela, et al.Bioorganic Chemistry|March 19, 2024
Investigation on production and reaction conditions of sucrose synthase based glucosylation cascade towards flavonoid modificationAgata Matera, Kinga Dulak, Hanna Werner, et al.Pageof 869