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Bioorganic Chemistry|March 26, 2026
Rational design and preclinical evaluation of 68Ga-labeled PEG-modified dimeric FAP radiotracersZehua Li, Yihao Feng, Hongrui Zhang, et al.Bioorganic Chemistry|April 19, 2026
DeepSAT-guided discovery of new eunicellin-type Diterpenoids from Cladiella krempfi and Sinularia ornataYi-Xian Qiu, Wei-Kang Xie, Sheng-Hui Zhu, et al.Bioorganic Chemistry|May 27, 2025
Structure activity relationship of Aristolochic acid analogues: Inhibitory effect on human and rat gonadal 3β-Hydroxysteroid dehydrogenasesWeijian Zhu, Zhuoqi Chen, Shaowei Wang, et al.Bioorganic Chemistry|May 27, 2025
An NTCP-mediated liver-targeting chimeras (NTLiverTac) design strategy and its application to hepatoblastoma modelsJing Liang, Weihong Luo, Wen Xu, et al.Bioorganic Chemistry|April 20, 2026
Design, synthesis, and biological evaluation of pyranone-carbamate hybrids as selective butyrylcholinesterase inhibitors with anti-neuroinflammatory activity for Alzheimer's diseaseXueyan Liu, Jiexin Xu, Chen Lin, et al.Bioorganic Chemistry|May 24, 2025
Investigating the multi-mechanistic anticancer effects of 4-bisarylurea thiouracil derivatives in breast cancer cellsMohamed Fares, Muhammad Alsherbiny, Islam A Elkelesh, et al.Bioorganic Chemistry|May 9, 2026
Cascade-driven β-Lapachone cycle in a photothermal/self-oxygenating MXene nanoplatform for synergistic tumor therapyDongmei Li, Mengqing Li, Qing He, et al.Bioorganic Chemistry|May 6, 2026
Donepezil-derived multi-target-directed ligands: design, synthesis, and anti-Alzheimer's evaluationMarwa S K Bassiouny, Mai I Shahin, Maiy Y Jaballah, et al.Bioorganic Chemistry|May 6, 2026
Exploration of novel costunolide derivatives bearing indole/indoline as anti-ulcerative colitis agents by targeting JAK2-STAT3 pathwaysHengli Yang, Yuan Jiang, Ruijuan Yang, et al.Bioorganic Chemistry|May 10, 2026
l-NBDNJ allosteric chaperone for multiple defective enzymes involved in lysosomal storage disorders (LSDs)Anna Esposito, Maria Stabile, Eliana De Gregorio, et al.Pageof 869