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Bioorganic Chemistry|August 8, 2026
Synthesis and evaluation of 3,5-disubstituted isothiazolo[4,5-b]pyridines, pyrazolo[4,3-b]pyridines and isothiazolo[3,4-b]pyrazines as inhibitors of PIKfyveLing-Jie Gao, Mathy Froeyen, Chieh-Wen Lo, et al.Bioorganic Chemistry|August 13, 2026
A dual-state emissive fluorescent probe for 2D and 3D intracellular picric acid sensingYu Lei, Zhiyong Ji, Wei Xiang, et al.Bioorganic Chemistry|August 17, 2026
Discovery and activity evaluation of fungal chitin synthase inhibitors via virtual screeningKun Gao, Xiaoyue Zhang, Wenjie Wang, et al.Bioorganic Chemistry|August 17, 2026
Lipoic acid-conjugated chalcones exert antitumor activity via ROS elevation and ferroptosisXinyue Bi, Haifu Sun, Kaihong Wang, et al.Bioorganic Chemistry|September 22, 2026
Design, synthesis, structure-activity relationship and in-silico studies of novel pyrazolo[1,5-a]pyrimidine derivatives as selective COX-2 inhibitors with promising anti-inflammatory activity and safety profileAlaa Omar Mohamed Helmy, Azza T Taher, Eman Z El Razaz, et al.Bioorganic Chemistry|September 22, 2026
FA1 site-targeted fluorescent probe for HSA detection and labeling: Biomedical applications and MD insights into local conformational perturbationJing Zhang, Jian-Heng Li, Xiu-Yuan Wu, et al.Bioorganic Chemistry|September 21, 2026
Photoinitiator based on oxime ester for photodynamic antibacterial therapy and wound healingZhihui Zhang, Yu Zhang, Bosong Zhou, et al.Bioorganic Chemistry|September 21, 2026
Novel L-Asparaginases from the human gut microbiome: Genome mining, biochemical characterization, and in vitro anti-leukemic activityDuygu Delican, Ozan Kılıçkaya, Ozkan Ozden, et al.Bioorganic Chemistry|September 23, 2026
Conventional and microwave-assisted synthesis of pyridine-linked 1,3,4-oxadiazole derivatives as promising antimicrobial agents: Structure-activity relationship and computational investigations using molecular docking, molecular dynamics simulation, MM-GBSA and DFTDarshan H Divetia, Devayat R Bhadarka, Vijay H Dodiya, et al.Bioorganic Chemistry|September 24, 2026
Azobenzene-bridged potent divalent ligands of Pseudomonas aeruginosa LecAYu Fan, Barbora Svomova, Martin Lepsik, et al.Pageof 869