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Bioorganic Chemistry|September 27, 2026
Diterpenoids from the leaves of Thuja orientalis L. and their inhibitory effects on PTP1B and α-glucosidaseThi Oanh Vu, Thi Nguyet Anh Dinh, Thi Ly Pham, et al.Bioorganic Chemistry|October 2, 2026
A lysosome-targeted dual-lock fluorescent probe based on synergistic pH/viscosity response for visualizing autophagy and tumor tissuesYaqiong Kong, Rong Wu, Lehua Cheng, et al.Bioorganic Chemistry|October 2, 2026
Design, synthesis and anticancer potential of new peptide conjugates via urokinase inhibition: biological and in silico studiesTaghreed Abdelstar Sheha, Amany S Mostafa, Shahenda M El-Messery, et al.Bioorganic Chemistry|October 18, 2026
Anti-HIV-1 activity and mechanism of action of homoplantaginin: A multitarget flavonoid compoundXin Liu, Qiuzhen Qin, Jie Liu, et al.Bioorganic Chemistry|October 20, 2026
Design, synthesis, and pharmacological evaluation of 7-substituted 1,2,4-triazolo[1,5-a]pyrimidine derivatives as novel antiepileptic lead candidates targeting Nav1.2 channelsLuqian He, Qiaoliang Zhang, Wenjuan Ma, et al.Bioorganic Chemistry|October 23, 2026
Modulation of strain-selective antimicrobial activity by the supramolecular ensemble of a pillar[5]arene with a proteaseVildan Sultanaev, Anastasia Nazarova, Igor Sedov, et al.Bioorganic Chemistry|October 27, 2026
Ligulaplenolides A-S, nineteen undescribed eremophilane-type sesquiterpenoids from Ligularia platyglossa and their anti-inflammatory activityXiao-Song Zhu, Qiong Wang, Tian-Rong Yang, et al.Bioorganic Chemistry|October 26, 2026
Novel NIR DDNP-type solvatochromic and fluorogenic probes for amyloid β detectionMatic Rogan, Lana Blinc, Luka Rejc, et al.Bioorganic Chemistry|October 28, 2026
C-4-functionalized cyclogeraniols from saffron: Structural diversity, Enantiomerism, and stereochemistry-dependent anti-melanogenic activityTing-Ting Li, Si-Bo Ji, Si-Qi Ma, et al.Bioorganic Chemistry|October 28, 2026
Discovery of novel pyridine-2-tetrazole derivatives as in vivo memory enhancement agentsNguyen Viet Hung, Van-Hai Hoang, Le Thien Bao Long, et al.Pageof 869