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Bioorganic Chemistry|September 7, 2019
Synthesis, in-vitro cholinesterase inhibition, in-vivo anticonvulsant activity and in-silico exploration of N-(4-methylpyridin-2-yl)thiophene-2-carboxamide analogsGulraiz Ahmad, Nasir Rasool, Komal Rizwan, et al.Bioorganic Chemistry|September 7, 2019
Design and evaluation of non-carboxylate 5-arylidene-2-thioxo-4-imidazolidinones as novel non-competitive inhibitors of protein tyrosine phosphatase 1BRosaria Ottanà, Paolo Paoli, Giulia Lori, et al.Bioorganic Chemistry|August 31, 2019
Pyrazole[3,4-d]pyridazine derivatives: Molecular docking and explore of acetylcholinesterase and carbonic anhydrase enzymes inhibitors as anticholinergics potentialsParham Taslimi, Fikret Türkan, Adnan Cetin, et al.Bioorganic Chemistry|September 3, 2019
Synthesis, anticancer activity and molecular docking studies on 1,2-diarylbenzimidazole analogues as anti-tubulin agentsYa-Liang Zhang, Rong Yang, Lin-Ying Xia, et al.Bioorganic Chemistry|September 4, 2019
Xanthones from the stems of Cudrania tricuspidata and their inhibitory effects on pancreatic lipase and fat accumulationYang Hee Jo, Seon Beom Kim, Jong Hoon Ahn, et al.Bioorganic Chemistry|September 14, 2019
Design, synthesis, and biological evaluation of novel dual FFA1 (GPR40)/PPARδ agonists as potential anti-diabetic agentsZheng Li, Lijun Hu, Xuekun Wang, et al.Bioorganic Chemistry|September 14, 2019
Promising antibacterial agents against multidrug resistant Staphylococcus aureusSrikanth Gatadi, Y V Madhavi, Sidharth Chopra, et al.Bioorganic Chemistry|September 14, 2019
Tyrosinase inhibitory effects of Vinca major and its secondary metabolites: Enzyme kinetics and in silico inhibition model of the metabolites validated by pharmacophore modellingSuat Sari, Burak Barut, Arzu Özel, et al.Bioorganic Chemistry|September 17, 2019
Novel [1,2,4]triazolo[1,5-a]pyrimidine derivatives as potent antitubulin agents: Design, multicomponent synthesis and antiproliferative activitiesFang Yang, Liang-Zhentian Yu, Peng-Cheng Diao, et al.Bioorganic Chemistry|August 3, 2019
Sulfonamides incorporating piperazine bioisosteres as potent human carbonic anhydrase I, II, IV and IX inhibitorsNiccolò Chiaramonte, Silvia Bua, Andrea Angeli, et al.Pageof 864