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Bioorganic Chemistry|November 4, 2020
New methyl 5-(halomethyl)-1-aryl-1H-1,2,4-triazole-3-carboxylates as selective COX-2 inhibitors and anti-inflammatory agents: Design, synthesis, biological evaluation, and docking studySin-Min Li, Shuo-En Tsai, Chia-Yin Chiang, et al.Bioorganic Chemistry|November 4, 2020
Prenylated xanthones and benzophenones from the fruits of Garcinia bracteata and their potential antiproliferative and anti-inflammatory activitiesQing Xue, Yu Chen, Huijun Yin, et al.Bioorganic Chemistry|November 4, 2020
Discovery of novel artemisinin-sulfonamidehybrids as potential carbonicanhydraseIX inhibitors with improved antiproliferative activitiesRan An, Bin Lin, Shuang Zhao, et al.Bioorganic Chemistry|November 4, 2020
Evaluation and comparison of the commonly used bioassays of human indoleamine 2,3-dioxygenase 1 (IDO1) and tryptophan 2,3-dioxygenase (TDO)Shengnan Zhang, Leilei Guo, Dan Yang, et al.Bioorganic Chemistry|November 4, 2020
Design, synthesis and antitumor evaluation of novel 5-methylpyrazolo[1,5-a]pyrimidine derivatives as potential c-Met inhibitorsGuolin Luo, Yanxia Ma, Xintong Liang, et al.Bioorganic Chemistry|November 4, 2020
Fungal mediated biotransformation of melengestrol acetate, and T-cell proliferation inhibitory activity of biotransformed compoundsSaira Javed, Atia-Tul-Wahab, Almas Jabeen, et al.Bioorganic Chemistry|November 16, 2020
Synthesis of triphenylphosphonium dibenzothiophene S-oxide derivatives and their effect on cell cycle as photodeoxygenation-based cytotoxic agentsAnkita Isor, Austin T O'Dea, John T Petroff, et al.Bioorganic Chemistry|November 16, 2020
Flavonoids from Barnebydendron riedelii leaf extract mitigate thioacetamide-induced hepatic encephalopathy in rats: The interplay of NF-κB/IL-6 and Nrf2/HO-1 signaling pathwaysSara M Baraka, Dalia O Saleh, Neveen S Ghaly, et al.Bioorganic Chemistry|February 15, 2020
NMR for screening and a biochemical assay: Identification of new FPPS inhibitors exerting anticancer activityManuela Grimaldi, Rosario Randino, Elena Ciaglia, et al.Bioorganic Chemistry|February 17, 2020
Arylidenes of Quinolin-2-one scaffold as Erlotinib analogues with activities against leukemia through inhibition of EGFR TK/ STAT-3 pathwaysMohammed A I Elbastawesy, Mohamed Ramadan, Yaseen A M M El-Shaier, et al.Pageof 865