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Bioorganic Chemistry|November 23, 2021
Enhancing cofactor regeneration of cyanobacteria for the light-powered synthesis of chiral alcoholsJianhua Fan, Yinghui Zhang, Ping Wu, et al.Bioorganic Chemistry|December 24, 2021
Design and synthesis of ibuprofen-quinoline conjugates as potential anti-inflammatory and analgesic drug candidatesAmany M Ghanim, Adel S Girgis, Benson M Kariuki, et al.Bioorganic Chemistry|December 27, 2021
Anti-inflammatory, ulcerogenic and platelet activation evaluation of novel 1,4-diaryl-1,2,3-triazole neolignan-celecoxib hybridsJosyelen L Felipe, Tatiana B Cassamale, Leticia D Lourenço, et al.Bioorganic Chemistry|December 27, 2021
Utilization of cyanopyridine in design and synthesis of first-in-class anticancer dual acting PIM-1 kinase/HDAC inhibitorsAmr K A Bass, El-Shimaa M Nageeb, Mona S El-Zoghbi, et al.Bioorganic Chemistry|December 27, 2021
Degrading FLT3-ITD protein by proteolysis targeting chimera (PROTAC)Yong Chen, Xue Yuan, Minghai Tang, et al.Bioorganic Chemistry|December 5, 2021
Click ferrocenyl-erlotinib conjugates active against erlotinib-resistant non-small cell lung cancer cells in vitroPrzemysław Biegański, Martina Godel, Chiara Riganti, et al.Bioorganic Chemistry|December 30, 2021
Design, synthesis, biological screening and molecular docking studies of novel multifunctional 1,4-di (aryl/heteroaryl) substituted piperazine derivatives as potential antitubercular and antimicrobial agentsBruktawit Mekonnen Sanka, Dereje Mamo Tadesse, Endale Teju Bedada, et al.Bioorganic Chemistry|October 27, 2022
HDAC/JAK dual target inhibitors of cancer-related targets: The success of nonclearable linked pharmacophore modeLiyun Zhao, Qi Liang, Ye He, et al.Bioorganic Chemistry|October 29, 2022
Identification of a novel nitroflavone-based scaffold for designing mutant-selective EGFR tyrosine kinase inhibitors targeting T790M and C797S resistance in advanced NSCLCMinnelli Cristina, Laudadio Emiliano, Sorci Leonardo, et al.Bioorganic Chemistry|November 6, 2022
Annulated pyrazole derivatives as a novel class of urokinase (uPA) inhibitors: Green synthesis, anticancer activity, DNA-damage evaluation, and molecular modelling studyPaula S Farag, Asmaa M AboulMagd, Magdy M Hemdan, et al.Pageof 866