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Bioorganic Chemistry|February 13, 2022
Lead optimization and biological evaluation of diazenylbenzenesulfonamides inhibitors against glyoxalase-I enzyme as potential anticancer agentsButhina A Al-Oudat, Nizar A Al-Shar'i, Qosay A Al-Balas, et al.Bioorganic Chemistry|October 3, 2021
Synthesis and biological evaluation of 2,5-diaryl-1,3,4-oxadiazole derivatives as novel Src homology 2 domain-containing protein tyrosine phosphatase 2 (SHP2) inhibitorsXiang-Dong Meng, Li-Xin Gao, Zhi-Jia Wang, et al.Bioorganic Chemistry|October 3, 2021
Synthesis, characterization and biological evaluation of indomethacin derived thioureas as purinergic (P2Y1, P2Y2, P2Y4, and P2Y6) receptor antagonistsSehrish Bano, Ghulam Shabir, Aamer Saeed, et al.Bioorganic Chemistry|October 7, 2021
Design, synthesis and mechanistic study of novel diarylpyrazole derivatives as anti-inflammatory agents with reduced cardiovascular side effectsNoha H Amin, Mohammed I A Hamed, Maha M Abdel-Fattah, et al.Bioorganic Chemistry|February 13, 2022
Discovery and structural optimization of 9-O-phenylsulfonyl-berberines as new lipid-lowering agentsYuan Kong, Yong-Jia Yi, Xiao-Qing Liu, et al.Bioorganic Chemistry|February 13, 2022
Interaction between CD44 and highly condensed hyaluronic acid through crosslinking with proteinsReika Tsuji, Soichi Ogata, Shinichi MochizukiBioorganic Chemistry|February 26, 2022
Discovery of new pyrimido[5,4-c]quinolines as potential antiproliferative agents with multitarget actions: Rapid synthesis, docking, and ADME studiesRamadan A Mekheimer, Samar M R Allam, Mariam A Al-Sheikh, et al.Bioorganic Chemistry|February 26, 2022
Revealing 2-dimethylhydrazino-2-alkyl alkynyl sphingosine derivatives as sphingosine kinase 2 inhibitors: Some hints on the structural basis for selective inhibitionMacarena Corro-Morón, Albert Granell, Varbina Ivanova, et al.Bioorganic Chemistry|April 30, 2019
Discovery of pyrazolopyrimidine derivatives as potent BTK inhibitors with effective anticancer activity in MCLFansheng Ran, Yang Liu, Meixia Liu, et al.Bioorganic Chemistry|April 17, 2019
Synthesis, antitumor testing and molecular modeling study of some new 6-substituted amido, azo or thioureido-quinazolin-4(3H)-onesMohamed A Sabry, Heba A Ewida, Ghada S Hassan, et al.Pageof 868