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European Journal of Medicinal Chemistry|December 31, 2017
Design, synthesis, and biological evaluation of polo-like kinase 1/eukaryotic elongation factor 2 kinase (PLK1/EEF2K) dual inhibitors for regulating breast cancer cells apoptosis and autophagyZhaoping Pan, Yujuan Chen, Jingyan Liu, et al.European Journal of Medicinal Chemistry|December 31, 2017
Synthesis and evaluation of 2-(3-arylureido)pyridines and 2-(3-arylureido)pyrazines as potential modulators of Aβ-induced mitochondrial dysfunction in Alzheimer's diseaseAhmed Elkamhawy, Jung-Eun Park, Ahmed H E Hassan, et al.European Journal of Medicinal Chemistry|October 10, 2017
4-Alkyliden-azetidinones modified with plant derived polyphenols: Antibacterial and antioxidant propertiesDaria Giacomini, Rosario Musumeci, Paola Galletti, et al.European Journal of Medicinal Chemistry|May 25, 2023
Proteolysis-targeting chimeras in biotherapeutics: Current trends and future applicationsQiong Li, Li Zhou, Siyuan Qin, et al.European Journal of Medicinal Chemistry|May 24, 2023
Synthesis and evaluation of DAG-lactone derivatives with HIV-1 latency reversing activityTakahiro Ishii, Takuya Kobayakawa, Kouki Matsuda, et al.European Journal of Medicinal Chemistry|May 26, 2023
Challenges for the development of mutant isocitrate dehydrogenases 1 inhibitors to treat gliomaQing-Xin Wang, Peng-Yu Zhang, Qing-Qing Li, et al.European Journal of Medicinal Chemistry|April 23, 2023
Discovery of ML210-Based glutathione peroxidase 4 (GPX4) degrader inducing ferroptosis of human cancer cellsHan Wang, Chao Wang, Bingru Li, et al.European Journal of Medicinal Chemistry|May 2, 2023
Biological activity of 1,2,3-triazole-2-amino-1,4-naphthoquinone derivatives and their evaluation as therapeutic strategy for malaria controlRenata Maria Costa Souza, Lilian Maria Lapa Montenegro Pimentel, Laryssa Kathleen Mendonça Ferreira, et al.European Journal of Medicinal Chemistry|March 30, 2023
Targeting the multifaceted neurotoxicity of Alzheimer's disease by tailored functionalisation of the curcumin scaffoldErsilia De Lorenzi, Francesca Seghetti, Andrea Tarozzi, et al.European Journal of Medicinal Chemistry|March 30, 2023
Targeting glutaminase 1 (GLS1) by small molecules for anticancer therapeuticsYangyang Chen, Lun Tan, Jing Gao, et al.Pageof 1,618