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Journal of Medicinal Chemistry|August 26, 2021
Discovery of First-in-Class Peptidomimetic Neurolysin Activators Possessing Enhanced Brain Penetration and StabilityMd Shafikur Rahman, Shikha Kumari, Shiva Hadi Esfahani, et al.
Journal of Medicinal Chemistry|August 12, 2021
Synthetic Glycolipids as Molecular Vaccine Adjuvants: Mechanism of Action in Human Cells and In Vivo ActivityFabio A Facchini, Alberto Minotti, Andrea Luraghi, et al.
Journal of Medicinal Chemistry|August 13, 2021
Discovery of ASTX029, A Clinical Candidate Which Modulates the Phosphorylation and Catalytic Activity of ERK1/2Tom D Heightman, Valerio Berdini, Luke Bevan, et al.
Journal of Medicinal Chemistry|August 20, 2021
1,3-Diarylpyrazolyl-acylsulfonamides as Potent Anti-tuberculosis Agents Targeting Cell Wall Biosynthesis in Mycobacterium tuberculosisLutete Peguy Khonde, Rudolf Müller, Grant A Boyle, et al.
Journal of Medicinal Chemistry|August 20, 2021
Pharmacophore-Based Design of Phenyl-[hydroxycyclohexyl] Cycloalkyl-Carboxamide Mitofusin Activators with Improved Neuronal ActivityXiawei Dang, Sidney B Williams, Sriram Devanathan, et al.
Journal of Medicinal Chemistry|August 3, 2021
Azide-Dye Unexpected Bone Targeting for Near-Infrared Window II Osteoporosis ImagingXiaoqing Zhang, Aiyan Ji, Zhiming Wang, et al.
Journal of Medicinal Chemistry|August 3, 2021
Are Pt(IV) Prodrugs That Release Combretastatin A4 True Multi-action Prodrugs?Claudia Schmidt, Tomer Babu, Hana Kostrhunova, et al.
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