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Journal of Medicinal Chemistry|October 27, 2015
Targeting Mitogen-Activated Protein Kinase-Activated Protein Kinase 2 (MAPKAPK2, MK2): Medicinal Chemistry Efforts To Lead Small Molecule Inhibitors to Clinical TrialsMario Fiore, Stefano Forli, Fabrizio ManettiJournal of Medicinal Chemistry|November 17, 2015
Discovery of 6-(4-{[5-Cyclopropyl-3-(2,6-dichlorophenyl)isoxazol-4-yl]methoxy}piperidin-1-yl)-1-methyl-1H-indole-3-carboxylic Acid: A Novel FXR Agonist for the Treatment of DyslipidemiaMichael J Genin, Ana B Bueno, Javier Agejas Francisco, et al.Journal of Medicinal Chemistry|November 18, 2015
Disrupting Acetyl-Lysine Recognition: Progress in the Development of Bromodomain InhibitorsF Anthony Romero, Alexander M Taylor, Terry D Crawford, et al.Journal of Medicinal Chemistry|November 18, 2015
Synthesis and Biological Activity of 2-Methylene Analogues of Calcitriol and Related CompoundsIzabela K Sibilska, Marcin Szybinski, Rafal R Sicinski, et al.Journal of Medicinal Chemistry|November 13, 2015
Discovery of Nanomolar Dengue and West Nile Virus Protease Inhibitors Containing a 4-Benzyloxyphenylglycine ResidueMira A M Behnam, Dominik Graf, Ralf Bartenschlager, et al.Journal of Medicinal Chemistry|November 14, 2015
Discovery of a First-in-Class, Potent, Selective, and Orally Bioavailable Inhibitor of the p97 AAA ATPase (CB-5083)Han-Jie Zhou, Jinhai Wang, Bing Yao, et al.Journal of Medicinal Chemistry|November 10, 2015
Discovery and Structure-Guided Optimization of Diarylmethanesulfonamide Disrupters of Glucokinase-Glucokinase Regulatory Protein (GK-GKRP) Binding: Strategic Use of a N → S (nN → σ*S-X) Interaction for Conformational ConstraintLewis D Pennington, Michael D Bartberger, Michael D Croghan, et al.Journal of Medicinal Chemistry|November 10, 2015
Pyrrolo[3,4-c]pyridine-1,3(2H)-diones: A Novel Antimycobacterial Class Targeting Mycobacterial RespirationRenier van der Westhuyzen, Susan Winks, Colin R Wilson, et al.Journal of Medicinal Chemistry|April 6, 2016
Biological Characterization and in Vivo Assessment of the Activity of a New Synthetic Macrocyclic Antifungal CompoundDavide Deodato, Giorgio Maccari, Filomena De Luca, et al.Journal of Medicinal Chemistry|April 6, 2016
Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Protein-Protein Interaction as a Target for Next-Generation Anti-influenza TherapeuticsSerena Massari, Laura Goracci, Jenny Desantis, et al.Pageof 3,137