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Journal of Medicinal Chemistry|July 23, 2015
Synthesis of Thrombolytic Sol-Gel Coatings: Toward Drug-Entrapped Vascular GraftsYulia Chapurina, Vasiliy V Vinogradov, Alexander V Vinogradov, et al.Journal of Medicinal Chemistry|June 5, 2015
Fragment-Based Design of Selective Nanomolar Ligands of the CREBBP BromodomainAndrea Unzue, Min Xu, Jing Dong, et al.Journal of Medicinal Chemistry|June 6, 2015
One-pot reaction to obtain N,N'-disubstituted guanidines of pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine scaffold as human A3 adenosine receptor antagonistsPier Giovanni Baraldi, Stefania Baraldi, Giulia Saponaro, et al.Journal of Medicinal Chemistry|June 11, 2015
Discovery of 1-{4-[3-fluoro-4-((3s,6r)-3-methyl-1,1-dioxo-6-phenyl-[1,2]thiazinan-2-ylmethyl)-phenyl]-piperazin-1-yl}-ethanone (GNE-3500): a potent, selective, and orally bioavailable retinoic acid receptor-related orphan receptor C (RORc or RORγ) inverse agonistBenjamin P Fauber, Olivier René, Yuzhong Deng, et al.Journal of Medicinal Chemistry|June 13, 2015
Benzoxaborole antimalarial agents. Part 4. Discovery of potent 6-(2-(alkoxycarbonyl)pyrazinyl-5-oxy)-1,3-dihydro-1-hydroxy-2,1-benzoxaborolesYong-Kang Zhang, Jacob J Plattner, Eric E Easom, et al.Journal of Medicinal Chemistry|June 13, 2015
Fragment-based exploration of binding site flexibility in Mycobacterium tuberculosis BioARan Dai, Todd W Geders, Feng Liu, et al.Journal of Medicinal Chemistry|June 19, 2015
Strategies for the Discovery of Target-Specific or Isoform-Selective ModulatorsPeng Zhan, Yukihiro Itoh, Takayoshi Suzuki, et al.Journal of Medicinal Chemistry|August 19, 2016
Synthesis and Biological Evaluation of N-[2-(4-Hydroxyphenylamino)-pyridin-3-yl]-4-methoxy-benzenesulfonamide (ABT-751) Tricyclic Analogues as Antimitotic and Antivascular Agents with Potent in Vivo Antitumor ActivityZacharie Segaoula, Julien Leclercq, Valérie Verones, et al.Journal of Medicinal Chemistry|August 19, 2016
Drug Discovery against Psoriasis: Identification of a New Potent FMS-like Tyrosine Kinase 3 (FLT3) Inhibitor, 1-(4-((1H-Pyrazolo[3,4-d]pyrimidin-4-yl)oxy)-3-fluorophenyl)-3-(5-(tert-butyl)isoxazol-3-yl)urea, That Showed Potent Activity in a Psoriatic Animal ModelGuo-Bo Li, Shuang Ma, Ling-Ling Yang, et al.Journal of Medicinal Chemistry|August 19, 2016
Purine-Type Compounds Induce Microtubule Fragmentation and Lung Cancer Cell Death through Interaction with KataninTing-Chun Kuo, Ling-Wei Li, Szu-Hua Pan, et al.Pageof 3,134