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Journal of Medicinal Chemistry|December 29, 2017
Systematic Tuning of Fluoro-galectin-3 Interactions Provides Thiodigalactoside Derivatives with Single-Digit nM Affinity and High SelectivityKristoffer Peterson, Rohit Kumar, Olof Stenström, et al.Journal of Medicinal Chemistry|March 9, 2018
Discovery of N1-(4-((7-Cyclopentyl-6-(dimethylcarbamoyl)-7 H-pyrrolo[2,3- d]pyrimidin-2-yl)amino)phenyl)- N8-hydroxyoctanediamide as a Novel Inhibitor Targeting Cyclin-dependent Kinase 4/9 (CDK4/9) and Histone Deacetlyase1 (HDAC1) against Malignant CancerYongtao Li, Xiaohe Luo, Qingxiang Guo, et al.Journal of Medicinal Chemistry|February 20, 2018
Structure-Based Optimization Strategies for G Protein-Coupled Receptor (GPCR) Allosteric Modulators: A Case Study from Analyses of New Metabotropic Glutamate Receptor 5 (mGlu5) X-ray StructuresJohn A Christopher, Zoltán Orgován, Miles Congreve, et al.Journal of Medicinal Chemistry|February 20, 2018
Synthesis and Biological Evaluation of ( E)-4-Hydroxy-3-methylbut-2-enyl Phosphate (HMBP) Aryloxy Triester Phosphoramidate Prodrugs as Activators of Vγ9/Vδ2 T-Cell Immune ResponsesMartin S Davey, Roshni Malde, Rory C Mykura, et al.Journal of Medicinal Chemistry|March 7, 2018
UNC-51-like Kinase 1: From an Autophagic Initiator to Multifunctional Drug TargetLan Zhang, Liang Ouyang, Yongzhi Guo, et al.Journal of Medicinal Chemistry|March 7, 2018
Synthesis and Biological Evaluation of Selenium-Containing 4-Anilinoquinazoline Derivatives as Novel Antimitotic AgentsBaijiao An, Bo Wang, Jinhui Hu, et al.Journal of Medicinal Chemistry|March 7, 2018
Discovery of Novel KRAS-PDEδ Inhibitors by Fragment-Based Drug DesignLong Chen, Chunlin Zhuang, Junjie Lu, et al.Journal of Medicinal Chemistry|February 16, 2018
Design, Synthesis, and Evaluation of a Novel Series of Indole Sulfonamide Peroxisome Proliferator Activated Receptor (PPAR) α/γ/δ Triple Activators: Discovery of Lanifibranor, a New Antifibrotic Clinical CandidateBenaïssa Boubia, Olivia Poupardin, Martine Barth, et al.Journal of Medicinal Chemistry|February 13, 2018
Monomeric and Dimeric 68Ga-Labeled Bombesin Analogues for Positron Emission Tomography (PET) Imaging of Tumors Expressing Gastrin-Releasing Peptide Receptors (GRPrs)Christos Liolios, Benjamin Buchmuller, Ulrike Bauder-Wüst, et al.Journal of Medicinal Chemistry|February 15, 2018
Exploiting the S4-S5 Specificity of Human Neutrophil Proteinase 3 to Improve the Potency of Peptidyl Di(chlorophenyl)-phosphonate Ester Inhibitors: A Kinetic and Molecular Modeling AnalysisCarla Guarino, Natalia Gruba, Renata Grzywa, et al.Pageof 3,134