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Pascal Heitel

8PUBLICATIONS
4CO-AUTHORS
Molecular medicineBiomolecular modelling and designCheminformatics and quantitative structure-activity relationshipsNutrigenomics and personalised nutritionProteins and peptides
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Journal

Publications (8)

Sort by Publication Date:
|Jun 05, 2026
Silymarin and Its Isolated Flavanonol Lignans Are Liver X Receptor Antagonists.

|Oct 23, 2025
Scaffold Fusion and SAR Transfer with a Chemical Language Model Generates Novel Liver X Receptor Modulators.

Nils Christiaan Bandomir, Tim Hörmann, Annette Kärcher

|Mar 19, 2024
Screening of Chelidonium majus isoquinoline alkaloids reveals berberine and chelidonine as selective ligands for the nuclear receptors RORβ and HNF4α, respectively.

Sohrab Salehi, Espen Schallmayer, Nils Bandomir

|Jan 27, 2023
A triple farnesoid X receptor and peroxisome proliferator-activated receptor α/δ activator reverses hepatic fibrosis in diet-induced NASH in mice.

Pascal Heitel, Giuseppe Faudone, Moritz Helmstädter

|Jan 21, 2023
Emerging TACnology: Heterobifunctional Small Molecule Inducers of Targeted Posttranslational Protein Modifications.

Pascal Heitel

|Jul 21, 2020
Design and Structural Optimization of Dual FXR/PPARδ Activators.

Simone Schierle, Sebastian Neumann, Pascal Heitel

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Frequent Collaborators

4 joint publications

Daniel Merk

1 joint publications

Ewgenij Proschak

1 joint publications

Apirat Chaikuad

1 joint publications

Stefan Knapp

Frequent Collaborators

4 joint publications

Daniel Merk

1 joint publications

Ewgenij Proschak

1 joint publications

Apirat Chaikuad

1 joint publications

Stefan Knapp