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Simone Brogi

60PUBLICATIONS
141CO-AUTHORS
Haematological tumoursCheminformatics and quantitative structure-activity relationshipsPredictive and prognostic markersMolecular targetsCancer therapy (excl. chemotherapy and radiation therapy)
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Journal

Publications (60)

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|Jul 04, 2026
Taginostat, a new quinolone-based HDAC6 inhibitor, promotes apoptosis of chronic lymphocytic leukemia cells in vitro and in vivo by activating STAT4.

|Jun 29, 2026
Integrated structure-based and fragment-guided design of isonicotinic acid derivatives as potential KDM4A inhibitors: an in silico study.

|Apr 24, 2026
Discovery of thieno[2,3-<i>d</i>]pyrimidine-based dual Aurora B/VEGFR-2 inhibitors with potent anticancer activity: molecular docking, mechanistic studies, and <i>in vivo</i> validation in a breast cancer model.

|Apr 06, 2026
Dimeric Anthraquinone Rugulosin A Induces Apoptosis in Lung Adenocarcinoma and Targets PI3K/AKT/MAPK Pathways <i>In Silico</i>.

Joe Anthony H Manzano, Elian Angelo M Abellanosa, Jose Paolo P Aguilar

|Mar 20, 2026
Second-generation prokineticin PKR<sub>1</sub> receptor agonists: Advancing cardioprotection against chemotherapy-induced toxicity.

Anais Audebrand, Simone Brogi, Mustafa Tezeren

|Feb 23, 2026
Quinazolinone-Based PqsR Modulators Suppress Quorum-Sensing-Driven Virulence in <i>Pseudomonas aeruginosa</i>.

Valeria Tudino, Marta Mellini, Leonardo Milioni

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Frequent Collaborators

18 joint publications

Sandra Gemma

16 joint publications

Stefania Butini

14 joint publications

Giuseppe Campiani

12 joint publications

Gabriele Carullo

6 joint publications

Hajar Sirous

5 joint publications

Vincenzo Calderone

4 joint publications

Anna Ramunno

4 joint publications

Nicola Relitti

4 joint publications

Stefano Federico

4 joint publications

Allan Patrick G Macabeo

Frequent Collaborators

18 joint publications

Sandra Gemma

16 joint publications

Stefania Butini

14 joint publications

Giuseppe Campiani

12 joint publications

Gabriele Carullo