Jenny Desantis

11PUBLICATIONS
21CO-AUTHORS
Biomolecular modelling and designProteins and peptidesMedical devicesPharmaceutical delivery technologiesMolecular targets
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Publications (11)

|Sep 13, 2024
Between Theory and Practice: Computational/Experimental Integrated Approaches to Understand the Solubility and Lipophilicity of PROTACs.

Andrea Venturi, Stefano Di Bona, Jenny Desantis

|Apr 11, 2024
Use of ionic liquids in amidation reactions for proteolysis targeting chimera synthesis.

Michela Eleuteri, Jenny Desantis, Gabriele Cruciani

|Sep 12, 2023
VHL-Modified PROteolysis TArgeting Chimeras (PROTACs) as a Strategy to Evade Metabolic Degradation in In Vitro Applications.

Beatrice Castellani, Michela Eleuteri, Stefano Di Bona

|Feb 27, 2023
MassChemSite for In-Depth Forced Degradation Analysis of PARP Inhibitors Olaparib, Rucaparib, and Niraparib.

Stefano Bonciarelli, Jenny Desantis, Simone Cerquiglini

|Nov 26, 2022
Exploiting ELIOT for Scaffold-Repurposing Opportunities: TRIM33 a Possible Novel E3 Ligase to Expand the Toolbox for PROTAC Design.

Tommaso Palomba, Giusy Tassone, Carmine Vacca

|Aug 31, 2022
PROTACs bearing piperazine-containing linkers: what effect on their protonation state?

Jenny Desantis, Andrea Mammoli, Michela Eleuteri

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