Henry I Mosberg
8PUBLICATIONS
2CO-AUTHORS
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Publications (8)
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|Dec 21, 2020
SAR Matrices Enable Discovery of Mixed Efficacy μ-Opioid Receptor Agonist Peptidomimetics with Simplified Structures through an Aromatic-Amine Pharmacophore.Sean Henry, Jessica P Anand, Ashley C Brinkel
|Jan 28, 2020
Aromatic-Amine Pendants Produce Highly Potent and Efficacious Mixed Efficacy μ-Opioid Receptor (MOR)/δ-Opioid Receptor (DOR) Peptidomimetics with Enhanced Metabolic Stability.Sean Henry, Jessica P Anand, Jack J Twarozynski
|Dec 18, 2019
Incorporation of Agouti-Related Protein (AgRP) Human Single Nucleotide Polymorphisms (SNPs) in the AgRP-Derived Macrocyclic Scaffold c[Pro-Arg-Phe-Phe-Asn-Ala-Phe-dPro] Decreases Melanocortin-4 Receptor Antagonist Potency and Results in the Discovery of Melanocortin-5 Receptor Antagonists.Zoe M Koerperich, Mark D Ericson, Katie T Freeman
|Jun 15, 2019
Novel Dimethyltyrosine-Tetrahydroisoquinoline Peptidomimetics with Aromatic Tetrahydroisoquinoline Substitutions Show in Vitro Kappa and Mu Opioid Receptor Agonism.Deanna Montgomery, Jessica P Anand, Nicholas W Griggs
|Mar 30, 2019
Structural Simplification of a Tetrahydroquinoline-Core Peptidomimetic μ-Opioid Receptor (MOR) Agonist/δ-Opioid Receptor (DOR) Antagonist Produces Improved Metabolic Stability.Sean P Henry, Thomas J Fernandez, Jessica P Anand
|Mar 28, 2019
Dual Pharmacophores Explored via Structure-Activity Relationship (SAR) Matrix: Insights into Potent, Bifunctional Opioid Ligand Design.Anthony F Nastase, Jessica P Anand, Aaron M Bender
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