Mizuki Takahashi

4PUBLICATIONS
11CO-AUTHORS
Cheminformatics and quantitative structure-activity relationshipsEnvironment policyMolecular targets
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Publications (4)

|Dec 18, 2023
A covalent fragment-based strategy targeting a novel cysteine to inhibit activity of mutant EGFR kinase.

Naoki Kuki, David L Walmsley, Kazuo Kanai

|Dec 26, 2022
Discovery of DS-9300: A Highly Potent, Selective, and Once-Daily Oral EP300/CBP Histone Acetyltransferase Inhibitor.

Ryutaro Kanada, Yoshiko Kagoshima, Takashi Suzuki

|Jul 28, 2019
Preclinical Development of U3-1784, a Novel FGFR4 Antibody Against Cancer, and Avoidance of Its On-target Toxicity.

René Bartz, Keisuke Fukuchi, Toshiaki Ohtsuka

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