Élie Besserer-Offroy

11PUBLICATIONS
39CO-AUTHORS
Proteins and peptidesToxicology (incl. clinical toxicology)Signal transductionInnate immunityCheminformatics and quantitative structure-activity relationships
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Publications (11)

|Dec 12, 2025
Structure-based design of macrocyclic peptides to generate functional antibodies against G protein-coupled receptors.

Marie-Edith Nepveu-Traversy, Malihe Hassanzadeh, Laurent Bruneau-Cossette

|Apr 01, 2025
Opioid Analgesics: Rise and Fall of Ligand Biased Signaling and Future Perspectives in the Quest for the Holy Grail.

Émile Breault, Rebecca L Brouillette, Terence E Hébert

|Mar 10, 2022
Monitoring TRPC7 Conformational Changes by BRET Following GPCR Activation.

Cécile Pétigny, Audrey-Ann Dumont, Hugo Giguère

|May 21, 2021
Structural insights on ligand recognition at the human leukotriene B4 receptor 1.

Nairie Michaelian, Anastasiia Sadybekov, Élie Besserer-Offroy

|Dec 08, 2020
Structure-Based Virtual Screening of Ultra-Large Library Yields Potent Antagonists for a Lipid GPCR.

Arman A Sadybekov, Rebecca L Brouillette, Egor Marin

|Dec 08, 2019
Structural basis of ligand selectivity and disease mutations in cysteinyl leukotriene receptors.

Anastasiia Gusach, Aleksandra Luginina, Egor Marin

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