Gianni Chessari
10PUBLICATIONS
38CO-AUTHORS
Get your video featured.
Publish with JoVEGet your video featured.
Publish with JoVE
Publications (10)
Sort by Publication Date:
|Apr 09, 2026
From KRASG12D to Pan-KRAS Inhibitors─A Journey Enabled by Synthetic Innovation and Structure-Based Drug Design.Xiaoshen Ma, David L Sloman, Timothy J Henderson
|Jun 27, 2024
Fragment-Based Discovery of a Series of Allosteric-Binding Site Modulators of β-Glucocerebrosidase.Nick Palmer, Christopher Agnew, Caroline Benn
|Mar 11, 2024
Fragment-Based Discovery of Allosteric Inhibitors of SH2 Domain-Containing Protein Tyrosine Phosphatase-2 (SHP2).James E H Day, Valerio Berdini, Joan Castro
|Dec 18, 2023
Enabling synthesis in fragment-based drug discovery (FBDD): microscale high-throughput optimisation of the medicinal chemist's toolbox reactions.Chloe Townley, Davide Branduardi, Gianni Chessari
|May 30, 2023
Accelerated Chemical Reaction Optimization Using Multi-Task Learning.Connor J Taylor, Kobi C Felton, Daniel Wigh
|Sep 14, 2022
X-ray Screening of an Electrophilic Fragment Library and Application toward the Development of a Novel ERK 1/2 Covalent Inhibitor.Jeffrey D St Denis, Gianni Chessari, Anne Cleasby
Pageof 2
Frequent Collaborators
6 joint publications
Christopher N Johnson
4 joint publications
Jeffrey D St-Denis
4 joint publications
Benjamin D Cons
3 joint publications
Christopher C F Hamlett
3 joint publications
John W Liebeschuetz
3 joint publications
Amanda Price
3 joint publications
Rachel Grainger
3 joint publications
Rhian S Holvey
3 joint publications
David G Twigg
3 joint publications
Paul N Mortenson
