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Gordon J Lockbaum

14PUBLICATIONS

25CO-AUTHORS

Molecular targetsProteins and peptidesAutonomic nervous systemPharmacogenomicsCheminformatics and quantitative structure-activity relationships

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Publications (14)

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|Nov 19, 2025

Discovery of Kinesin KIF18A Inhibitor ATX020: Tactical Application of Silicon Atom Replacement.

Brian A Sparling, Hyelee Lee, Mary-Margaret Zablocki

|Apr 29, 2025

Discovery of ATX968: An Orally Available Allosteric Inhibitor of DHX9.

Matthew H Daniels, Jennifer Castro, Young-Tae Lee

|Apr 09, 2025

Characterization of exoribonuclease XRN1 as a cancer target and identification of adenosine-3',5'-bisphosphate as a potent enzyme inhibitor.

Gordon J Lockbaum, Maureen M Lynes, Sophie A Shen

|Nov 10, 2022

Dual Inhibitors of Main Protease (M<sup>Pro</sup>) and Cathepsin L as Potent Antivirals against SARS-CoV2.

Santanu Mondal, Yongzhi Chen, Gordon J Lockbaum

|Jun 21, 2022

Defining the substrate envelope of SARS-CoV-2 main protease to predict and avoid drug resistance.

Ala M Shaqra, Sarah N Zvornicanin, Qiu Yu J Huang

|Sep 10, 2021

Pan-3C Protease Inhibitor Rupintrivir Binds SARS-CoV-2 Main Protease in a Unique Binding Mode.

Gordon J Lockbaum, Mina Henes, Jeong Min Lee

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Frequent Collaborators

11 joint publications

Celia A Schiffer

10 joint publications

Nese Kurt Yilmaz

6 joint publications

Akbar Ali

3 joint publications

Robert A Copeland

3 joint publications

Serena J Silver

3 joint publications

Kenneth W Duncan

3 joint publications

Brian A Sparling

2 joint publications

Jennifer Timm

2 joint publications

Paul R Thompson

2 joint publications

Young-Tae Lee

Frequent Collaborators

11 joint publications

Celia A Schiffer

10 joint publications

Nese Kurt Yilmaz

6 joint publications

Akbar Ali

3 joint publications

Robert A Copeland

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