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Síntesis enantioselectiva de la (+) -cefalostatina 1 y 1

Kevin C Fortner1, Darryl Kato, Yoshiki Tanaka

  • 1Department of Chemistry and Chemical Biology, Harvard University, 12 Oxford Street, Cambridge, Massachusetts 02138, USA.

Journal of the American Chemical Society
|December 9, 2009
PubMed
Resumen

Este estudio presenta una nueva síntesis enantioselectiva de la cefalostatina 1. El método utiliza estrategias únicas de oxidación, hidroxilación C-H y ciclización para la construcción eficiente de compuestos.

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