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Updated: Nov 26, 2025

Preparation of 6-aminocyclohepta-2,4-dien-1-one Derivatives via Tricarbonyltroponeiron
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Síntesis directa de 2-azidoaminas no protegidas a partir de alquenos a través de una reacción de difuncionalización

Szabolcs Makai1, Eric Falk1, Bill Morandi1

  • 1ETH Zürich, Vladimir-Prelog-Weg 3, HCI, 8093 Zürich, Switzerland.

Journal of the American Chemical Society
|December 10, 2020
PubMed
Resumen

Desarrollamos un sencillo método catalizado por el hierro para sintetizar 2-azidoaminas a partir de alquenos. Estos compuestos son precursores clave de las diaminas vicinales, cruciales en las moléculas biológicamente activas y el descubrimiento de fármacos.

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