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Updated: Jul 15, 2026

Drug-induced Sensitization of Adenylyl Cyclase: Assay Streamlining and Miniaturization for Small Molecule and siRNA Screening Applications
09:39

Drug-induced Sensitization of Adenylyl Cyclase: Assay Streamlining and Miniaturization for Small Molecule and siRNA Screening Applications

Published on: January 27, 2014

アデニリルサイクラスによる信号開始と終了の促進

K Scholich1, J B Mullenix, C Wittpoth

  • 1Department of Pharmacology, University of Tennessee, Health Science Center, 874 Union Avenue, Memphis, TN 38163, USA.

Science (New York, N.Y.)
|February 26, 1999
PubMed
まとめ

アデニリルサイクラスは,GsalphaのGTPase活性化タンパク質 (GAP) として作用し,Gタンパク質の無活性化を加速します. また,受容体シグナル伝達を強化し,より迅速な細胞応答を促進します.

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