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Updated: Jul 26, 2026

Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
10:17

Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones

Published on: February 7, 2019

サイクロペプチドアルカロイドへの収束的アプローチ:サンジョイニンG1の全合成

Taoues Temal-Laïb1, Jacqueline Chastanet, Jieping Zhu

  • 1Institut de Chimie des Substances Naturelles, CNRS, 91198 Gif-sur-Yvette, France.

Journal of the American Chemical Society
|January 24, 2002
PubMed
まとめ

研究者は,アリル-アルキルエーテル結合を持つサイクロペプチドアルカロイドの新合成を,分子内S(N) Ar反応を用いて開発した. この方法により,天然産物サンジョイニンG1. 1を合成することが成功しました.

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