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Updated: Jul 17, 2026

A Two-Step Protocol for Umpolung Functionalization of Ketones Via Enolonium Species
08:12

A Two-Step Protocol for Umpolung Functionalization of Ketones Via Enolonium Species

Published on: August 16, 2018

ベータアミノアルコールを供給するヒドロキシケトンの反選択的直接触媒非対称マンニッヒ型反応

Shigeki Matsunaga1, Naoya Kumagai, Shinji Harada

  • 1Graduate School of Pharmaceutical Sciences, The University of Tokyo, Hongo, Bunkyo-ku, Tokyo 113-0033, Japan.

Journal of the American Chemical Society
|April 17, 2003
PubMed
まとめ

この研究では,抗ベータアミノアルコールを合成するための新しい触媒法が導入されています. このプロセスは,新しい触媒システムを使用して,高収量と優れたステレオ選択性を達成します.

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