関連する実験動画

Updated: Jul 6, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

レチノイドX受容体の反応経路を選択するレチノイド

J M Lehmann1, L Jong, A Fanjul

  • 1Cancer Center, La Jolla Cancer Research Foundation, La Jolla, CA 92037.

Science (New York, N.Y.)
|December 18, 1992
PubMed
まとめ

新しいレチノイドは,レチノイドX受容体 (RXRs) ホモダイマーを,レチノ酸受容体 (RARs) に独立して選択的に活性化します. これにより,異なるレチノイドシグナル伝達経路の独立した活性化が可能になります.

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