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Updated: Jul 17, 2026

Protein WISDOM: A Workbench for In silico De novo Design of BioMolecules
10:58

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Published on: July 25, 2013

タンパク質キナーゼ阻害剤:構造から薬物設計への洞察

Martin E M Noble1, Jane A Endicott, Louise N Johnson

  • 1Laboratory of Molecular Biophysics, Department of Biochemistry, Rex Richards Building, University of Oxford, Oxford 3X2 3QU, UK.

Science (New York, N.Y.)
|March 20, 2004
PubMed
まとめ

このレビューは,臨床用キナーゼ阻害剤を,利用可能な構造データで取り上げ,がんや炎症などの疾患における薬物設計と阻害機構におけるその役割を強調しています.

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