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Updated: Aug 23, 2026

A Microwave-Assisted Direct Heteroarylation of Ketones Using Transition Metal Catalysis
07:06

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Published on: February 16, 2020

Et2Zn/リンクされた-BINOL複合体を用いた水素キセトンの直接触媒非対称マニッヒ型反応:抗または合成β-アミノアルコールの合成

Shigeki Matsunaga1, Takamasa Yoshida, Hiroyuki Morimoto

  • 1Graduate School of Pharmaceutical Sciences, The University of Tokyo, Hongo, Bunkyo-ku, Tokyo 113-0033, Japan.

Journal of the American Chemical Society
|July 15, 2004
PubMed
まとめ

この研究では,亜鉛結合BINOL複合体を用いた直接触媒非対称マニッヒ型反応の詳細が示されています. この反応は,イミン保護基を調整することによって,高ステレオ選択性を持つ抗またはシンベータアミノアルコールを効率的に生成します.

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