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Updated: Jul 15, 2026

Split-and-pool Synthesis and Characterization of Peptide Tertiary Amide Library
13:37

Split-and-pool Synthesis and Characterization of Peptide Tertiary Amide Library

Published on: June 20, 2014

フォルマミシンの全合成

Timothy B Durham1, Nicolas Blanchard, Brad M Savall

  • 1Department of Chemistry, University of Michigan, 930 North University, Ann Arbor, Michigan 48109, USA.

Journal of the American Chemical Society
|July 30, 2004
PubMed
まとめ

研究者は,細胞毒性のある天然産物であるホルマミシンのエナンチオセレクティブ・トータル合成を達成しました. 重要なステップには,アセタル形成,スズキ結合,およびこの複雑な分子のためのステレオ選択的グリコシデーションが含まれています.

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