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Updated: Jul 20, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

物質P (NK1) 受容体の強力なノンペプチドアンタゴニストである

R M Snider1, J W Constantine, J A Lowe

  • 1Department of Exploratory Medicinal Chemistry, Central Research Division, Pfizer Inc., Groton, CT 06340.

Science (New York, N.Y.)
|January 25, 1991
PubMed
まとめ

CP-96,345は,物質P (NK1) 受容体の選択的ノンペプチドアンタゴニストである. この化合物は,物質Pの結合とその効果をin vivoで効果的にブロックし,物質Pの研究に貴重なツールを提供します.

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