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Updated: Jul 6, 2026

Constructing Cyclic Peptides Using an On-Tether Sulfonium Center
07:11

Constructing Cyclic Peptides Using an On-Tether Sulfonium Center

Published on: September 28, 2022

アニオンテンプレート反応による擬似ペプチドマクロサイクルのモジュール合成のための超分子制御

Ignacio Alfonso1, Michael Bolte, Miriam Bru

  • 1Departamento de Química Orgánica Biológica, Instituto de Investigaciones Químicas y Ambientales de Barcelona, Consejo Superior de Investigaciones Científicas, Jordi Girona, 18-26, E-08034, Barcelona, Spain. iarqob@iiqab.csic.es

Journal of the American Chemical Society
|April 12, 2008
PubMed
まとめ

アニオンテンプレート合成により,シドオペプチドマクロサイクルが効率的に生成されます. このワンポット・ツーステップ・リダクティブ・アミネーション・メソッドは,アニオンテンプレートを用いてマクロサイクライゼーションを誘導し,安定したテトラアミンのマクロサイクルを生成します.

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