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Updated: Jul 5, 2026

Preparation of N-(2-alkoxyvinyl)sulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
10:42

Preparation of N-(2-alkoxyvinyl)sulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines

Published on: January 3, 2018

代替ピリジンの単純なモジュール合成です

Songbai Liu1, Lanny S Liebeskind

  • 1Department of Chemistry, Emory University, 1515 Dickey Drive, Atlanta, Georgia 30322, USA.

Journal of the American Chemical Society
|May 10, 2008
PubMed
まとめ

新しいモジュラー法では,銅で触媒化されたカスケード反応を使用して,高度に置換されたピリジンを合成します. この効率的なプロセスは,クロスカップリング,電循環,空気酸化を含み,ピリジンを良好な量から優れた量まで生成します.

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Basicity of Heterocyclic Aromatic Amines

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Arenediazonium substitution reactions occur when the diazonium group is substituted by various functional groups such as halides, hydroxyl, nitrile, etc. For instance, arenediazonium salts react with copper(I) salts of chloride, bromide, or cyanide to form corresponding aryl chlorides, bromides, and nitriles. These reactions are named Sandmeyer reactions. Although the mechanism of this reaction is complicated, as illustrated in Figure 1, they are believed to progress via an aryl copper...
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