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Updated: Jul 3, 2026

Preparation of Contiguous Bisaziridines for Regioselective Ring-Opening Reactions
04:38

Preparation of Contiguous Bisaziridines for Regioselective Ring-Opening Reactions

Published on: July 28, 2022

アジリジンによるエナンチオおよびダイアステロ選択的触媒性アルキル化反応

Thomas A Moss1, David R Fenwick, Darren J Dixon

  • 1School of Chemistry, The University of Manchester, Oxford Road, Manchester M13 9PL, UK.

Journal of the American Chemical Society
|July 12, 2008
PubMed
まとめ

この研究では,N-スルフォニルアジリジンを用いた最初の非対称な相移転触媒アルキル化が導入されました. この方法は,高エナチオ選択性を持つ有価なアミノエチレン製品を効率的に生成し,非対称合成を推進します.

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