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Updated: Jun 22, 2026

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
07:30

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

Published on: January 21, 2020

局所生成のN-カルバモイルニトロンによる有機触媒的非対称形式 [3 + 2] サイクル添加

Claudio Gioia1, Francesco Fini, Andrea Mazzanti

  • 1Department of Organic Chemistry A. Mangini, University of Bologna, viale Risorgimento 4, 40136 Bologna, Italy.

Journal of the American Chemical Society
|June 26, 2009
PubMed
まとめ

この研究は,N-BocとN-Cbzで保護されたイソキザゾリジンを合成するための新しい有機触媒反応を導入します. この方法は,容易に入手可能な触媒を使用し,高収量と純度で貴重な化学的構成要素を提供します.

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