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Updated: May 1, 2026

Protocol for the Synthesis of Ortho-trifluoromethoxylated Aniline Derivatives
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パラジアム触媒による非活性アルケンの分子内アミノフッ素化

Tao Wu1, Guoyin Yin, Guosheng Liu

  • 1State Key Laboratory of Organometallics Chemistry, Shanghai Institute of Organic Chemistry, Chinese Academy of Science, 354 Fenglin Road, Shanghai, China, 200032.

Journal of the American Chemical Society
|October 28, 2009
PubMed
まとめ

研究者らは,活性化されていないアルケーンから近隣のフッ素アミンを生成するための新しいパラジウム触媒反応を開発した. この方法は,銀フッ化物 (AgF) と高価ヨウ素反応剤を使用し,C-F結合形成において高い地域選択性を達成します.

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