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Updated: Jun 11, 2026

Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
10:17

Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones

Published on: February 7, 2019

C-nor-D-ホモステロイドに対するバイオミメティックアプローチ

Philipp Heretsch1, Sebastian Rabe, Athanassios Giannis

  • 1Institut für Organische Chemie, Fakultät für Chemie und Mineralogie, Universität Leipzig, Johannisallee 29, D-04103 Leipzig, Germany.

Journal of the American Chemical Society
|July 6, 2010
PubMed
まとめ

研究者は,サイクロパミンなどの天然製品に不可欠なC-nor-D-ホモステロイドを合成するための3段階のバイオミメティック方法を開発しました. この効率的な戦略は,17-ケトステロイドでも機能し,幅広い適用性を提供します.

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