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Updated: Jun 10, 2026

Preparation and Delivery of Protein Microcrystals in Lipidic Cubic Phase for Serial Femtosecond Crystallography
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Preparation and Delivery of Protein Microcrystals in Lipidic Cubic Phase for Serial Femtosecond Crystallography

Published on: September 20, 2016

X線結晶学によって明らかにされたヒトβ2アドレナージック受容体の逆アゴニストとアンタゴニストの保存された結合モード

Daniel Wacker1, Gustavo Fenalti, Monica A Brown

  • 1Department of Molecular Biology, The Scripps Research Institute, La Jolla, California 92037, USA.

Journal of the American Chemical Society
|July 31, 2010
PubMed
まとめ

ベータ (((2) アドレナージック受容体 (ベータ (((2) AR) の構造研究により,異なる逆アゴニストおよびアンタゴニストと結合すると,局所的なわずかな変化が明らかになる. これらの発見は,薬物設計のためのリガンド相互作用を理解するのに役立ちます.

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Harvesting and Cryo-cooling Crystals of Membrane Proteins Grown in Lipidic Mesophases for Structure Determination by Macromolecular Crystallography18:45

Harvesting and Cryo-cooling Crystals of Membrane Proteins Grown in Lipidic Mesophases for Structure Determination by Macromolecular Crystallography

Published on: September 2, 2012

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