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Updated: Jun 3, 2026

Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles
11:45

Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles

Published on: August 22, 2018

置換されたパイペリジンの高度にダイアステロセレクティブのアリレーションです

Stephanie Seel1, Tobias Thaler, Keishi Takatsu

  • 1Department Chemie, Ludwig-Maximilians-Universität München, Butenandtstr. 5-13, Haus F, 81377 Munich, Germany.

Journal of the American Chemical Society
|March 11, 2011
PubMed
まとめ

新しい方法では,ネギシクロスカップリングを使用して,高いステレオ選択性を持つ代替パイペリジンを作成します. このアプローチは,シスまたはトランス同位体形成を制御し,ピペリジン合成の正確な制御を提供します.

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