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Updated: Jun 2, 2026

Methodology for Studying Interactions of Vitamin A Membrane Receptors and Opsin Protein with their Ligands in Generating the Retinylidene Protein
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Methodology for Studying Interactions of Vitamin A Membrane Receptors and Opsin Protein with their Ligands in Generating the Retinylidene Protein

Published on: October 4, 2024

14-epi-19-nortachysterolの開発と,ヒトのビタミンD受容体に対する前例のない結合構成

Daisuke Sawada1, Yuya Tsukuda, Hiroshi Saito

  • 1Faculty of Pharmaceutical Sciences, Teikyo University, 1091-1, Suwarashi, Sagamihara, Kanagawa 252-5195, Japan.

Journal of the American Chemical Society
|April 20, 2011
PubMed
まとめ

研究者らは新しい14-epi-19-nortachysterol誘導体を合成し,それらは安定し,ビタミンD受容体 (VDR) に強く結合することを発見しました. この研究は,ユニークな結合構成を持つ安定したタキステロール類の同類体を初めて分離したものです.

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