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Updated: May 25, 2026

Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles
11:45

Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles

Published on: August 22, 2018

ティオニウムイオンの誘発による中型環形成:アステリスクノリドDの全合成

Barry M Trost1, Aaron C Burns, Mark J Bartlett

  • 1Department of Chemistry, Stanford University, Stanford, California 94305-5080, USA. bmtrost@stanford.edu

Journal of the American Chemical Society
|January 13, 2012
PubMed
まとめ

研究者らは,自然産物であるアステリスクノリドDを初めて合成した. この9段階のプロセスは,ストレングマクロサイクルを効率的に作り,最も生物学的に活性な形態を生成しました.

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