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Updated: May 22, 2026

Protocol for the Synthesis of Ortho-trifluoromethoxylated Aniline Derivatives
08:43

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Published on: January 19, 2016

エナミドの非対称的な化:アニオニックキラル相転移触媒を用いてα-フッロアミンへのアクセス

Robert J Phipps1, Kenichi Hiramatsu, F Dean Toste

  • 1Department of Chemistry, University of California, Berkeley, 94720, United States.

Journal of the American Chemical Society
|May 12, 2012
PubMed
まとめ

チラルの相転移触媒は,Selectfluorを使用したエナミドのエナチオセレクティブ化を可能にします. この方法は,薬剤合成において決定的に重要なステレオ定義β-フッ素アミンの前駆体である有価なα-(フッ素) ベンゾイリミンへのアクセスを提供します.

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