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Updated: May 21, 2026

Inner Mitochondrial Membrane Sensitivity to Na+ Reveals Partially Segmented Functional CoQ Pools
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Published on: July 20, 2022

サイトクロームBC1複合体のピコモラーQ (o) サイト阻害剤の計算式発見

Ge-Fei Hao1, Fu Wang, Hui Li

  • 1Key Laboratory of Pesticide & Chemical Biology, Ministry of Education, College of Chemistry, Central China Normal University, Wuhan 430079, P. R. China.

Journal of the American Chemical Society
|June 14, 2012
PubMed
まとめ

フラグメントベース・ドラッグ・ディスカバリー (Fragment-based drug discovery, FBDD) は,現在,高通量メソッドを提供している. この新しいファーマコフォール関連仮想スクリーニング (PFVS) アプローチは,生体物理学的スクリーニングなしで強力な膜タンパク質阻害剤を特定します.

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