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Updated: May 19, 2026

A Two-Step Protocol for Umpolung Functionalization of Ketones Via Enolonium Species
08:12

A Two-Step Protocol for Umpolung Functionalization of Ketones Via Enolonium Species

Published on: August 16, 2018

銅で触媒化された非対称な分子内ウールマンC-N結合:インドリンのエナンチオセレクティブ製剤

Fengtao Zhou1, Jiajia Guo, Jianguang Liu

  • 1Key Laboratory of Regenerative Biology and Institute of Chemical Biology, Guangzhou Institutes of Biomedicine and Health, Chinese Academy of Sciences, No. 190 Kaiyuan Avenue, Guangzhou Science Park, Guangzhou 510530, China.

Journal of the American Chemical Society
|August 24, 2012
PubMed
まとめ

研究者は,最初のエナチオセレクティブの銅触媒ユルマンC-Nカップリングを開発しました. この方法では,高いエナチオメリック過剰を持つキラルインドリンとテトラヒドロキノリンを効率的に生成します.

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