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Updated: May 12, 2026

Constructing Cyclic Peptides Using an On-Tether Sulfonium Center
07:11

Constructing Cyclic Peptides Using an On-Tether Sulfonium Center

Published on: September 28, 2022

化学選択性セリン結合によるサイクリングによるダプトマイシン全合成

Hiu Yung Lam1, Yinfeng Zhang, Han Liu

  • 1Department of Chemistry, The University of Hong Kong, Pokfulam Road, Hong Kong, People's Republic of China.

Journal of the American Chemical Society
|April 9, 2013
PubMed
まとめ

研究者らは,新しい抗生物質であるダプトマイシンの完全な合成を達成しました. この画期的な発見により,ダプトマイシンアナログの作成が可能になり,新しい薬の開発のための構造-活性関係を探求することができます.

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