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Updated: May 7, 2026

Synthesis of a Borylated Ibuprofen Derivative Through Suzuki Cross-Coupling and Alkene Boracarboxylation Reactions
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Published on: November 30, 2022

サルフェン酸をアリルボロン酸とベンゾキサボロールで捕獲する

C Tony Liu1, Stephen J Benkovic

  • 1Department of Chemistry, Pennsylvania State University , University Park, Pennsylvania 16802, United States.

Journal of the American Chemical Society
|September 21, 2013
PubMed
まとめ

ベンゾキサボロールのようなボロン基化合物は,生物学的プロセスにおける重要な調節体であるシステイン-硫黄酸を捕まえます. この研究は,この修飾されたシステインを必要とする酵素を阻害することによって,その可能性を実証しています.

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