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Updated: Apr 26, 2026

A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

Published on: January 21, 2020

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4-ニトロピラゾリジンの触媒的非対称合成:光学的に活性な1,2,3-トリアミンへのアクセス

Lennart Lykke1, Bjørn Dreiø Carlsen, Raoní Scheibler Rambo

  • 1Center for Catalysis, Department of Chemistry, Aarhus University , DK-8000 Aarhus C, Denmark.

Journal of the American Chemical Society
|July 30, 2014
PubMed
まとめ

この研究は,4-ニトロピラゾリジンの最初の触媒的非対称合成を導入しています. この方法は,3つのステレオセンターを持つ光学的に活性な化合物を生成し,1,2,3-トリアミンを生成するのに役立ちます.

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